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Agile Bioanalytical Services CRO

Inquire Now About Our 20+ Years Discovery DMPK & ADME Services At FDA Audited Bioanalytical Lab

Accelerate Your Discovery DMPK & ADME Service!

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    • Cross-Species Microsomal, Hepatocyte, Plasma Stability For Diverse Modalities
    • Regulatory-Grade DDI With 7-Isoform CYP Inhibition, CYP Induction, PPB, Transporter Panels
    • Caco-2, MDCK-MDR1, PAMPA Permeability With Efflux Ratios To Flag P-gp Substrates
    • PhD-Led Met ID Or Soft-Spot Analysis On HRMS And HPLC-MS/MS With ~2-3 Week Turnaround

Regulated And Inspected By:

20+ Years Of Bioanalysis
700+ Small/Large Molecule Studies
500+ Custom Bioanalytical Assays
200+ Investigational Drugs
1,000+ Biomarker & Cytokine Assays

From Discovery Through IND - In Vitro ADME, DMPK & Met ID Services For Small Molecules, Biologics, Peptides

Microsomal Stability

Test compound depletion measured by LC-MS/MS for intrinsic clearance and half-life

Hepatocyte Stability

Cross-species hepatocyte incubations for intrinsic clearance, t½, metabolic soft spots

CYP Induction Assay

Cryopreserved human hepatocytes with mRNA fold-change and EC50 reporting across AhR, CAR, PXR

CYP Inhibition Assay

7-isoform IC50 panel and time-dependent IC50 shift in pooled human liver microsomes for DDI risk

Metabolite Identification

Identification and characterization of drug metabolites using high-resolution mass spectrometry

Plasma Protein Binding

Fraction unbound across species using rapid equilibrium dialysis

Permeability Assays

Apparent permeability and efflux ratios to flag P-gp substrates

Transporter Assays

DDI risk via MDR1, BCRP, OATP1B1/1B3, OAT1/3, OCT2, MATE1/2-K, BSEP substrate/inhibition

Don’t Wait, Start Your Drug Metabolism and Pharmacokinetics (ADME) Today!

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100+ Biotechs. 500+ Custom Assays. One Agile, FDA-Inspected ADME Services CRO.

Head, Bioanalytical Development

NorthEast BioLab goes the extra mile. We look forward to more meaningful collaborations

Sr. Dir., Bioanalytical Dev & QC

NorthEast BioLab offers a science-based, hands-on approach to the latest bioanalytical platforms

VP, Bioanalytical Development

NorthEast BioLab is the most responsive and thorough bioanalysis lab services CRO

VP, Development Operations

NorthEast BioLab’s scientists deliver high-quality data on time and within budget

VP, Biomarker Development

NorthEast BioLab is a responsive, collaborative, and reliable partner

Executive Director, Pharmacokinetics

We trust NorthEast BioLab to design and execute streamlined, impactful bioanalytical projects

Not Ready For Quote? Book 20-Min DMPK/ADME Services Call.

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